Researcher
Olivier Van Der Poorten
- Keywords:Chemistry (incl. biochemistry)
Affiliations
- Chemistry (Department)
Member
From8 Apr 2019 → 30 Sep 2021 - Faculty of Sciences and Bioengineering Sciences (Faculty)
Member
From6 Aug 2015 → 29 Mar 2018 - Chemistry (Department)
Member
From1 Oct 2013 → 3 Jun 2019 - Faculty of Sciences and Bioengineering Sciences (Faculty)
Member
From27 Jul 2011 → 5 Jul 2013
Projects
1 - 2 of 2
- Constrained tryptophan-based oligomers for intracellular and CNS drug delivery.From1 Oct 2018 → 3 Jun 2019Funding: FWO fellowships
- Conformationally tightened amino acids for peptide turn mimetics and drug transportFrom1 Jan 2014 → 31 Dec 2017Funding: IWT personal funding - strategic basic research grants
Publications
1 - 10 of 11
- 3-Substituted 2-isocyanopyridines as versatile convertible isocyanides for peptidomimetic design(2021)
Authors: Charlie Hollanders, Mathias Elsocht, Olivier Van der Poorten, Mouhamad Jida, Evelien Renders, Bert U. W. Maes, S Ballet
Pages: 6863-6866 - Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure †(2020)
Authors: Charlotte Martin, Luis E. Gimenez, Savannah Y. Williams, Yu Jing, Yiran Wu, Charlie Hollanders, Olivier Van der Poorten, S Gonzalez, K Van Holsbeeck, Santo Previti, et al.
Pages: 357-369 - Elucidating the active delta-opioid receptor crystal structure with peptide and small-molecule agonists(2019)
Authors: Tobias Claff, Jing Yu, Veronique Blais, Nilkanth Patel, Charlotte Martin, Lijie Wu, Gye Won Han, Brian J. Holleran, Olivier Van der Poorten, Kate L. White, et al.
- Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds. IF 2.593(2018)
Authors: Olivier Van der Poorten, Baptiste Legrand, Lubomir L. Vezenkov, Julia Garcia-Pindado, Nadir Bettache, Astrid Knuhtsen, Daniel Sejer Pedersen, Macarena Sanchez-Navarro, Jean Martinez, Meritxell Teixido, et al.
Pages: 696-705 - Rapid construction of substituted 3-amino-1,5-benzothiazepin-4(5H)-one dipeptide scaffolds through an Ugi-4CR - Ullmann cross-coupling sequence. IF 3.49(2018)
Authors: Olivier Van der Poorten, Robin Van Den Hauwe, Charlie Hollanders, Dirk Tourwé, Mouhamad Jida, S Ballet
Pages: 1242-1246 - Efficient One-Pot Access to Trisubstituted 2-Benzazepin-3-ones as Constrained Pseudopeptide Analogues and Privileged Scaffolds. IF 2.53(2018)
Authors: Olivier Van der Poorten, Mouhamad Jida, Dirk Tourwé, S Ballet
Pages: 400-408 - χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds. IF 3.794(2017)
Authors: Olivier Van der Poorten, Robin Van Den Hauwe, Emilie Eiselt, Cecilia Betti, Karel Jules Guillemyn, Nga N. Chung, François Hallé, Frédéric Bihel, Peter W. Schiller, Dirk Tourwé, et al.
Pages: 1177-1182 - Side Chain Cyclized Aromatic Amino Acids: Great Tools as Local Constraints in Peptide and Peptidomimetic Design. IF 6.259(2016)
Authors: Olivier Van der Poorten, Astrid Knuhtsen, Daniel Sejer Pedersen, S Ballet, Dirk Tourwé
Pages: 10865-10890 - Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases. IF 5.317(2016)
Authors: Astrid Knuhtsen, Baptiste Legrand, Olivier Van der Poorten, Muriel Amblard, Jean Martinez, S Ballet, Jesper L. Kristensen, Daniel Sejer Pedersen
Pages: 14022-14028 - T3P-promoted, mild one-pot syntheses of constrained polycyclic lactam dipeptide analogues via stereoselective Pictet-Spengler and Meyers’ lactamization reactions. IF 6.732(2015)
Authors: Mouhamad Jida, Olivier Van der Poorten, Karel Jules Guillemyn, Zofia Urbanczyk-Lipkowska, Dirk Tourwé, S Ballet
Pages: 4482-4485